Ceriscoides turgida (Roxb.) Tirveng. (syn. Gardenia turgida), a prominent member of the Rubiaceae family, is a deciduous medicinal tree traditionally valued across the Indian subcontinent for its diverse therapeutic properties. This review synthesizes current knowledge regarding the phytochemical profile, extraction methodologies, and biological activities of C. turgida roots. Phytochemical investigations reveal a rich reservoir of secondary metabolites, including triterpenoids, saponins, flavonoids, and phenolics. Comparative analysis of extraction techniques indicates that Soxhlet extraction using polar solvents like methanol provides superior yields of these metabolites compared to cold maceration, although maceration better preserves heat-sensitive antioxidants.